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Serotonin

Serotonin, also known as 5-hydroxytryptamine or 5-HT, is an organic monoamine neurotransmitter and hormone involved in a wide range of physiological processes. It is synthesized from the essential amino acid tryptophan by the enzymes tryptophan hydroxylase and aromatic L-amino acid decarboxylase. In humans, most 5-HT is produced outside the brain, in enterochromaffin cells of the gut, and stored in platelets; a smaller amount is produced in neurons of the raphe nuclei and functions as a neurotransmitter in the central nervous system. Because serotonin cannot cross the blood–brain barrier in meaningful amounts, peripheral and central serotonin operate largely in separate pools.

In the brain, serotonin modulates mood, emotion, sleep, appetite, cognition, and thermoregulation. In the periphery, it

Serotonin acts on a family of receptors designated 5-HT1 through 5-HT7, with at least several subtypes in

Disrupted serotonergic signaling is linked to mood and anxiety disorders. Pharmacological strategies include selective serotonin reuptake

regulates
gastrointestinal
motility,
vascular
tone,
and
hemostasis,
and
may
influence
wound
healing.
Release
from
neurons
is
calcium-dependent
and
terminated
primarily
by
reuptake
through
the
serotonin
transporter
(SERT).
Within
cells,
monoamine
oxidase
A
(MAO-A)
deaminates
serotonin
to
5-hydroxyindoleacetic
acid
(5-HIAA),
which
is
excreted
in
urine.
each
family.
5-HT3
is
a
ligand-gated
ion
channel;
the
others
are
G-protein-coupled
receptors.
Receptor
subtypes
mediate
diverse
effects;
for
example,
5-HT1A
receptors
are
involved
in
anxiolytic
and
antidepressant
mechanisms,
while
5-HT2A/2C
receptors
are
associated
with
mood
regulation
and
the
pharmacology
of
certain
psychedelic
drugs.
inhibitors
(SSRIs),
serotonin-norepinephrine
reuptake
inhibitors
(SNRIs),
and
other
agents
that
modulate
serotonin
levels.
Triptans
target
5-HT1B/1D
receptors
for
migraine
treatment,
and
psychedelics
act
on
5-HT2A
receptors.
Serotonin
syndrome
is
a
potential
risk
when
serotonergic
activity
is
excessively
increased.