Peksumasin
Peksumasin is a synthetic opioid analgesic developed by the pharmaceutical company Pfizer. It is a mu-opioid receptor agonist, meaning it binds to the mu-opioid receptors in the brain to produce its analgesic effects. Peksumasin was initially developed as a potential treatment for chronic pain, but it was later found to have a high potential for abuse and dependence, similar to other opioids. Due to these concerns, Pfizer discontinued the development of peksumasin in 2010. The drug was never marketed or approved for use in humans. Peksumasin is a member of the benzomorphan class of opioids, which are characterized by their unique chemical structure and their ability to bind to the mu-opioid receptor with high affinity. The development of peksumasin was part of a broader effort by Pfizer to discover new opioid analgesics with improved safety profiles. However, the company ultimately decided to focus on other areas of research and development. Peksumasin is not currently available for purchase or use, and its development has been discontinued.