Myokardielt
Myokardielt is a synthetic opioid analgesic developed by the pharmaceutical company Pfizer. It is a prodrug of myokardin, a potent mu-opioid receptor agonist. Myokardielt is designed to be rapidly converted into myokardin in the body, allowing for rapid onset of analgesic effects. It is used for the management of moderate to severe pain, including postoperative pain and cancer pain. The drug is typically administered orally, although it can also be given intravenously for more rapid onset of action. Myokardielt is available under the brand name Eltropy. The drug was approved by the U.S. Food and Drug Administration (FDA) in 2016 for the management of moderate to severe pain in adults. Common side effects of myokardielt include nausea, vomiting, constipation, and dizziness. Serious side effects can include respiratory depression, seizures, and allergic reactions. Myokardielt should be used with caution in patients with a history of opioid dependence or abuse, as well as those with respiratory depression or other serious medical conditions. It is important to note that myokardielt is a controlled substance in many countries due to its potential for abuse and dependence. As with all opioid analgesics, myokardielt should be used under the supervision of a healthcare provider and only when other non-opioid pain medications are not effective.